Microwave-Induced Synthesis of Enantiopure β- Lactams

Indrani B, Fredrick FB and

Abstract

Synthesis of enantiopure C-3/C-4 disubstituted β-lactams has been achieved through Staudinger cycloaddition reaction of acid chloride and imine under microwave irradiation. Importantly, reactions has been manipulated by proper selection of substrates to obtain both enantiomers in high yield.

Relevant Publications in Modern Chemistry & Applications